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10.1155/2022/7655033 26 Czarnecka-ChrebelskaK

Tan et al., reported that FIIN-2, an irreversible covalent FGFR inhibitor, formed the covalent binding mode at the Cys477 residue of FGFR4 in the DGF-out conformation (96)

& Wu, J

Takahashi M, Dillon TJ, Liu C, Kariya Y, Wang Z, Stork PJ